(3-トリフルオロメチルフェニル)(2-アミノ-4-メチル-5-メチル-3-チエニル)ケトン 化學特性,用途語,生産方法
使用
PD 81,723 is an allosteric potentiator that increases the functional effects of adenosine and adenosine analogs.
生物活性
Allosteric potentiator at the adenosine A 1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t 1/2 of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A 1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo .
(3-トリフルオロメチルフェニル)(2-アミノ-4-メチル-5-メチル-3-チエニル)ケトン 上流と下流の製品情報
原材料
準備製品