Omarigliptin (MK-3102)
|
- $55 - $5576
- Product name: Omarigliptin (MK-3102)
- CAS: 1226781-44-7
- MF: C17H20F2N4O3S
- MW: 398.43
- EINECS:682-558-0
- MDL Number:MFCD22573261
- Synonyms:(2R,3S,5R)-2-(2,5-difluorophenyl)-5-(2-(Methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-aMine;MK-3012;(2S,3R,5S)-2-(2,5-Difluorophenyl)-5-[2-(Methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-2H-pyran-3-aMine (MK-3102 enantioMer);(2R,3S,5R)-2-(2,5-Difluorophenyl)-5-[2-(methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-2H-pyran-3-amine;OMarigliptin (MK-3102);2R,3S,5R)-2-(2,5-Difluorophenyl)-5-[2-(methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-2H-pyran-3-amine MK3102;MK-3102 - M10588;MK-3102, >=98%
32 prices
Selected condition：
Brand
- AK Scientific
- Ambeed
- ApexBio Technology
- Arctom
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Matrix Scientific
- Medical Isotopes, Inc.
- TRC
Package
- 1mg
- 2mg
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- 1000mg
- ManufacturerAK Scientific
- Product number9051AF
- Product descriptionOmarigliptin
- Packaging2mg
- Price$158
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA115550
- Product descriptionOmarigliptin 98+%
- Packaging2mg
- Price$83
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA115550
- Product descriptionOmarigliptin 98+%
- Packaging5mg
- Price$149
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA115550
- Product descriptionOmarigliptin 98+%
- Packaging10mg
- Price$194
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA115550
- Product descriptionOmarigliptin 98+%
- Packaging50mg
- Price$328
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA115550
- Product descriptionOmarigliptin 98+%
- Packaging1g
- Price$5576
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB5868
- Product descriptionMK3102
- Packaging50mg
- Price$640
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS437410
- Product descriptionOmarigliptin ≥98%
- Packaging5mg
- Price$148
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181402
- Product descriptionMK-3102 (Omarigliptin ) >98%
- Packaging100mg
- Price$569.5
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181402
- Product descriptionMK-3102 (Omarigliptin ) >98%
- Packaging250mg
- Price$765
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181402
- Product descriptionMK-3102 (Omarigliptin ) >98%
- Packaging1000mg
- Price$1431.4
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number21454
- Product descriptionMK-3102 ≥98%
- Packaging1mg
- Price$57
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number21454
- Product descriptionMK-3102 ≥98%
- Packaging5mg
- Price$220
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number21454
- Product descriptionMK-3102 ≥98%
- Packaging10mg
- Price$395
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number21454
- Product descriptionMK-3102 ≥98%
- Packaging25mg
- Price$885
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-3948
- Product descriptionOmarigliptin
- Packaging2mg
- Price$55
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 9051AF | Omarigliptin | 2mg | $158 | 2021-12-16 | Buy |
| Ambeed | A115550 | Omarigliptin 98+% | 2mg | $83 | 2021-12-16 | Buy |
| Ambeed | A115550 | Omarigliptin 98+% | 5mg | $149 | 2021-12-16 | Buy |
| Ambeed | A115550 | Omarigliptin 98+% | 10mg | $194 | 2021-12-16 | Buy |
| Ambeed | A115550 | Omarigliptin 98+% | 50mg | $328 | 2021-12-16 | Buy |
| Ambeed | A115550 | Omarigliptin 98+% | 1g | $5576 | 2021-12-16 | Buy |
| ApexBio Technology | B5868 | MK3102 | 50mg | $640 | 2021-12-16 | Buy |
| Arctom | AS437410 | Omarigliptin ≥98% | 5mg | $148 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181402 | MK-3102 (Omarigliptin ) >98% | 100mg | $569.5 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181402 | MK-3102 (Omarigliptin ) >98% | 250mg | $765 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181402 | MK-3102 (Omarigliptin ) >98% | 1000mg | $1431.4 | 2021-12-16 | Buy |
| Cayman Chemical | 21454 | MK-3102 ≥98% | 1mg | $57 | 2024-03-01 | Buy |
| Cayman Chemical | 21454 | MK-3102 ≥98% | 5mg | $220 | 2024-03-01 | Buy |
| Cayman Chemical | 21454 | MK-3102 ≥98% | 10mg | $395 | 2024-03-01 | Buy |
| Cayman Chemical | 21454 | MK-3102 ≥98% | 25mg | $885 | 2024-03-01 | Buy |
| ChemScene | CS-3948 | Omarigliptin | 2mg | $55 | 2021-12-16 | Buy |
Properties
Boiling point :529.4±60.0 °C(Predicted)
Density :1.61±0.1 g/cm3(Predicted)
storage temp. :2-8°C(protect from light)
solubility :insoluble in EtOH; insoluble in H2O; ≥17.15 mg/mL in DMSO
form :solid
pka :9.11±0.60(Predicted)
color :White to off-white
InChI :InChI=1S/C17H20F2N4O3S/c1-27(24,25)23-7-10-6-22(8-16(10)21-23)12-5-15(20)17(26-9-12)13-4-11(18)2-3-14(13)19/h2-4,7,12,15,17H,5-6,8-9,20H2,1H3/t12-,15+,17-/m1/s1
InChIKey :MKMPWKUAHLTIBJ-ISTRZQFTSA-N
SMILES :[C@H]1(C2=CC(F)=CC=C2F)OC[C@H](N2CC3=CN(S(C)(=O)=O)N=C3C2)C[C@@H]1N
CAS DataBase Reference :1226781-44-7
Density :1.61±0.1 g/cm3(Predicted)
storage temp. :2-8°C(protect from light)
solubility :insoluble in EtOH; insoluble in H2O; ≥17.15 mg/mL in DMSO
form :solid
pka :9.11±0.60(Predicted)
color :White to off-white
InChI :InChI=1S/C17H20F2N4O3S/c1-27(24,25)23-7-10-6-22(8-16(10)21-23)12-5-15(20)17(26-9-12)13-4-11(18)2-3-14(13)19/h2-4,7,12,15,17H,5-6,8-9,20H2,1H3/t12-,15+,17-/m1/s1
InChIKey :MKMPWKUAHLTIBJ-ISTRZQFTSA-N
SMILES :[C@H]1(C2=CC(F)=CC=C2F)OC[C@H](N2CC3=CN(S(C)(=O)=O)N=C3C2)C[C@@H]1N
CAS DataBase Reference :1226781-44-7
Safety Information
| Symbol(GHS): |
|
|||||||||||||||||||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Signal word: | Warning | |||||||||||||||||||||||||||||||||||
| Hazard statements: |
|
|||||||||||||||||||||||||||||||||||
| Precautionary statements: |
|
Description
Merck earned its first global approval for omarigliptin in Japan in 2015, and phase III development is ongoing in other countries around the globe for this interesting small molecule DPP-4 inhibitor. Interestingly, while most DPP-4 inhibitors used to treat type 2 DM require daily administration, omarigliptin is a weekly treatment. The process-scale synthesis of omarigliptin has been nicely described in an October 2015 paper from the Merck process group.Related product price
- tert-butyl [(2R,3S)-2-(2,5-difluorophenyl)-5-hydroxytetrahydro-2H-pyran-3-yl]carbaMate
$55-941 - Alogliptin benzoate
$49-1871.1 - 221176-49-4
$310-1490
Suppliers and manufacturers
Capot Chemical Co.,Ltd.
Beijing Cooperate Pharmaceutical Co.,Ltd
Henan Tianfu Chemical Co.,Ltd.
Shanghai Yingrui Biopharma Co., Ltd.
ATK CHEMICAL COMPANY LIMITED
Lianyungang happen teng technology co., LTD
