Rp-cAMPS triethylammonium salt NEW
| Price | $489 | $2058 |
| Package | 1mg | 5mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-04-28 |
Product Details
| Product Name: Rp-cAMPS triethylammonium salt | CAS No.: 151837-09-1 |
| Supply Ability: 10g | Release date: 2025/04/28 |
Product Introduction
Bioactivity
| Name | Rp-cAMPS triethylammonium salt |
| Description | Rp-cAMPS triethylammonium salt is a competitive inhibitor of cAMP-dependent protein kinases I and II, inhibiting cAMP-induced conformational changes to block PKA activation. |
| In vitro | Rp-cAMPS triethylammonium salt inhibits CAMP-induced CAMP-dependent protein kinase I and II activation with Ki values of 12.5 μM and 4.5 μM. Rp-cAMPS triethylammonium salt (100 μM) reduced K+ current induced by calcitonin gene-related peptide (CGRP) in porcine smooth muscle cells. [2] |
| In vivo | Rp-cAMPS triethylammonium salt (10 μM, 15 min) reduced monosynaptic EPSCs of PB-CeLC and BLA-CeLC synapses in arthritic rats, but had no effect on control neurons in normal animals. [1] Intrabla infusion of Rp-cAMPS triethylammonium salt after cocaine memory reconsolidation impaired subsequent cocaine-seeking behavior in a dose-dependent, site-specific, and memory-reactivation dependent manner. [3] |
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | DMSO : 8 mg/mL (17.92 mM), Sonication is recommended. |
| Keywords | RpcAMPS triethylammonium salt | Rp-cAMPS triethylammonium | Rp cAMPS triethylammonium salt | PKA II | PKA I |
| Inhibitors Related | Daphnetin | Capivasertib | Ellagic acid | GSK180736A | Acefylline | Ro-3306 | Metadoxine | Staurosporine | 8-Bromo-cAMP sodium salt | Bucladesine sodium | Fasudil hydrochloride | JAK1/2/3 Inhibitor 1 |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, USA
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