Pentoxyverine NEW
| Price | $43 |
| Package | 1mL |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-06-13 |
Product Details
| Product Name: Pentoxyverine | CAS No.: 77-23-6 |
| Purity: 97.11% | Supply Ability: 10g |
| Release date: 2025/06/13 |
Product Introduction
Bioactivity
| Name | Pentoxyverine |
| Description | Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor, which causes alveolar relaxation and thus symptomatic relief. |
| In vitro | Pentoxyverine binds human σ? receptors with moderate affinity (Ki ~100-300 nM) and activates typical σ?-mediated cellular responses such as calcium flux[1]. |
| In vivo | Pentoxyverine (30-60 mg/kg, i.p.) exhibits antinociceptive effects in mice in thermal and inflammatory pain models. Pentoxyverine's effects are σ? receptor-dependent, as shown by partial reversal with σ? antagonist BD1047[1]. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice./Shipping at ambient temperature. |
| Solubility Information | DMSO : 200.00 mg/mL (599.75 mM), Sonication is recommended. |
| Keywords | Pentoxyverine |
| Inhibitors Related | Adiphenine hydrochloride | (+)-Sparteine | Pilocarpine nitrate | Clozapine N-Oxide | Urethane | Ribavirin | D-Menthol | Amitriptyline hydrochloride | Choline chloride | Propoxur | Pempidine | Otilonium bromide |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, USA
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