3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester
- CAS No.
- 1014691-61-2
- Chemical Name:
- 3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester
- Synonyms
- CS-738;GSK 0660;GSK-0660, >=98%;GSK-0660 (GSK0660);GSK0660 >=98% (HPLC);GSK0660, 10 mM in DMSO;GSK-0660;GSK 0660;GSK0660;GSK 0660, PPARdelta antagonist;4-Chloro-3-iodo-2,3-dihydro-1H-pyrrolo[2,3-b]pyridine;METHYL 3-[(4-ANILINO-2-METHOXYPHENYL)SULFAMOYL]THIOPHENE-2-CARBOXYLATE
- CBNumber:
- CB12518768
- Molecular Formula:
- C19H18N2O5S2
- Molecular Weight:
- 418.49
- MDL Number:
- MFCD12828770
- MOL File:
- 1014691-61-2.mol
- MSDS File:
- SDS
3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester Properties
Boiling point | 608.1±65.0 °C(Predicted) |
---|---|
Density | 1.413±0.06 g/cm3(Predicted) |
storage temp. | 2-8°C |
solubility | DMSO: soluble10mg/mL, clear |
form | powder |
pka | 8.51±0.50(Predicted) |
color | white to beige |
InChIKey | NDFKBGWLUHKMFY-UHFFFAOYSA-N |
UNSPSC Code | 12352203 |
NACRES | NA.77 |
3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester price More Price(30)
Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|---|
Sigma-Aldrich | G5797 | GSK0660 ≥98% (HPLC) | 1014691-61-2 | 5mg | $153 | 2022-05-15 | Buy |
Cayman Chemical | 15272 | GSK0660 ≥95% | 1014691-61-2 | 5mg | $97 | 2024-03-01 | Buy |
Cayman Chemical | 15272 | GSK0660 ≥95% | 1014691-61-2 | 10mg | $182 | 2024-03-01 | Buy |
Cayman Chemical | 15272 | GSK0660 ≥95% | 1014691-61-2 | 25mg | $427 | 2024-03-01 | Buy |
Cayman Chemical | 15272 | GSK0660 ≥95% | 1014691-61-2 | 50mg | $711 | 2024-03-01 | Buy |
3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester Chemical Properties,Uses,Production
Uses
GSK0660 has been used to study the effects of bezafibrate (BZA) on hypertrophy.
Definition
ChEBI: 3-[(4-anilino-2-methoxyphenyl)sulfamoyl]-2-thiophenecarboxylic acid methyl ester is a sulfonamide.
General Description
GSK0660 has antiangiogenic property in oxygen-induced retinopathy. It also regulates tumor necrosis factor-α (TNFα)-induced inflammation in human retinal microvascular endothelial cells (HRMECs).
Biochem/physiol Actions
GSK0660 is a potent PPARβ/δ antagonist with a pIC50 of 6.8 (160 nM). GSK0660 is nearly inactive on PPARα and PPARγ with IC50s greater than 10 μM.
storage
Store at +4°C
3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester Preparation Products And Raw materials
Raw materials
Preparation Products
Supplier | Tel | Country | ProdList | Advantage | |
---|---|---|---|---|---|
ATK CHEMICAL COMPANY LIMITED | +undefined-21-51877795 | ivan@atkchemical.com | China | 33024 | 60 |
career henan chemical co | +86-0371-86658258 +8613203830695 | factory@coreychem.com | China | 29807 | 58 |
TargetMol Chemicals Inc. | +17819995354 | marketing@targetmol.com | United States | 32295 | 58 |
Zhejiang J&C Biological Technology Co.,Limited | +1-2135480471 +1-2135480471 | sales@sarms4muscle.com | China | 10473 | 58 |
Alfa Chemistry | Info@alfa-chemistry.com | United States | 24072 | 58 | |
InvivoChem | +1-708-310-1919 +1-13798911105 | sales@invivochem.cn | United States | 6391 | 58 |
ShenZhen Trendseen Biological Technology Co.,Ltd. | 13417589054 | trendseenbio@gmail.com | China | 11681 | 58 |
Wuhan Topule Biopharmaceutical Co., Ltd | +8618327326525 | masar@topule.com | China | 8467 | 58 |
Aladdin Scientific | tp@aladdinsci.com | United States | 57505 | 58 | |
Amadis Chemical Company Limited | 571-89925085 | sales@amadischem.com | China | 131957 | 58 |
View Lastest Price from 3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester manufacturers
Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
---|---|---|---|---|---|---|---|---|
![]() |
2025-04-27 | GSK0660
1014691-61-2
|
US $39.00-106.00 / mg | 99.9% | 10g | TargetMol Chemicals Inc. | ||
![]() |
2019-12-24 | methyl 3-[(4-anilino-2-methoxyphenyl)sulfamoyl]thiophene-2-carboxylate
1014691-61-2
|
US $1.00 / KG | 1KG | Min98% HPLC | g/kg/ton | Career Henan Chemical Co |
-
- GSK0660
1014691-61-2
- US $39.00-106.00 / mg
- 99.9%
- TargetMol Chemicals Inc.
-
- methyl 3-[(4-anilino-2-methoxyphenyl)sulfamoyl]thiophene-2-carboxylate
1014691-61-2
- US $1.00 / KG
- Min98% HPLC
- Career Henan Chemical Co