Identification | Back Directory | [Name]
GP 2A | [CAS]
919077-81-9 | [Synonyms]
GP 2A CP 2A CB2 receptor agonist 3 CB2 receptor agonist 3,CB-2 receptor agonist 3 N-cyclohexyl-1-(2,4-dichlorophenyl)-6-methyl-4H-indeno[1,2-c]pyrazole-3-carboxamide N-CYCLOHEXYL-1-(2,4-DICHLOROPHENYL)-1,4-DIHYDRO-6-METHYLINDENO[1,2-C]PYRAZOLE-3-CARBOXAMIDE Indeno[1,2-c]pyrazole-3-carboxamide, N-cyclohexyl-1-(2,4-dichlorophenyl)-1,4-dihydro-6-methyl- | [Molecular Formula]
C24H23Cl2N3O | [MDL Number]
MFCD09971118 | [MOL File]
919077-81-9.mol | [Molecular Weight]
440.36 |
Hazard Information | Back Directory | [Uses]
GP 2A is a selective CB2 agonist that also shows modest agonism at CB1 receptors. | [Definition]
ChEBI: N-cyclohexyl-1-(2,4-dichlorophenyl)-6-methyl-4H-indeno[1,2-c]pyrazole-3-carboxamide is a member of pyrazoles and a ring assembly. | [Biological Activity]
Selective CB 2 receptor agonist; K i values are 7.6 and 900 nM for CB 2 and CB 1 receptors respectively. Increases P-ERK1/2 expression in HL-60 cells in vitro . |
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Company Name: |
BOC Sciences
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Tel: |
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Website: |
https://www.bocsci.com |
Company Name: |
Biorbyt Ltd.
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Tel: |
+44 (0)1223 859 353 |
Website: |
www.biorbyt.com |
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