Identification | Back Directory | [Name]
(3R)-1-[1-(anthracene-9-carbonyl)piperidin-4-yl]-N,N-diethylpiperidine-3-carboxamide | [CAS]
591778-83-5 | [Synonyms]
CP-610431 (3R)-1-[1-(anthracene-9-carbonyl)piperidin-4-yl]-N,N-diethylpiperidine-3-carboxamide | [Molecular Formula]
C30H37N3O2 | [MOL File]
591778-83-5.mol | [Molecular Weight]
471.634 |
Hazard Information | Back Directory | [Description]
CP-610431 is an isozyme-nonselective ACC inhibitor. CP-610431 inhibited ACC1 and ACC2 with IC50s of approximately 50 nm. Inhibition was reversible, uncompetitive with respect to ATP, and non-competitive with respect to bicarbonate, acetyl-CoA, and citrate, indicating interaction with the enzymatic carboxyl transfer reaction. |
|
|