Chemical Properties | Back Directory | [storage temp. ]
4°C, away from moisture | [solubility ]
DMSO : 200 mg/mL (388.72 mM; Need ultrasonic) | [form ]
Solid | [color ]
White to light yellow |
Hazard Information | Back Directory | [Biological Activity]
SETD2-IN-1 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. SETD2-IN-1 TFA has anti-proliferative effects[1]. | [References]
[1]. John Lampe, et al. Substituted indoles and methods of use thereof. WO2020037079A1. |
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