Chemical Properties | Back Directory | [Boiling point ]
620.5±55.0 °C(Predicted) | [density ]
1.30±0.1 g/cm3(Predicted) | [solubility ]
DMSO:20.83(Max Conc. mg/mL);57.0(Max Conc. mM) | [form ]
Solid | [pka]
14.62±0.50(Predicted) | [color ]
Light yellow to yellow |
Hazard Information | Back Directory | [Description]
GSK-3484862 is a non-covalent inhibitor for Dnmt1. GSK-3484862 induces DNA hypomethylation to against cancer. | [in vitro]
In total, methylation mapping supports the conclusion that GSK-3484862 treatment produces a drop in DNA methylation consistent with selective and near complete inhibition of DNMT1._x000D_
_x000D_
Reference: Epigenetics Chromatin. 2021 Dec 15;14(1):56. https://pubmed.ncbi.nlm.nih.gov/34906184/ | [target]
GSK-3484862 is a non-covalent inhibitor for DNA methyltransferase (Dnmt1). GSK-3484862 induces DNA hypomethylation to against cancer. |
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InvivoChem
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13549236410 |
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https://www.invivochem.cn/ |
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www.sangon.com |
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